Title

The Application Of Vinylogous Iminium Salt Derivatives To An Efficient Relay Synthesis Of The Pyrrole Containing Alkaloids Polycitone A And B

Keywords

Marine natural product; Pyrrole; Vinamidinium salt

Abstract

A new and efficient relay synthesis of the marine natural products polycitone A and B is described. The new strategy relies on the formation of 2,4-disubstituted pyrroles from a vinamidinium salt followed by electrophilic substitution at the 5-position of the pyrrole and Suzuki coupling at the 4-position to produce the tetrasubstituted heterocycle efficiently and with complete control of regiochemistry. © 2004 Elsevier Ltd. All rights reserved.

Publication Date

2-14-2005

Publication Title

Tetrahedron

Volume

61

Issue

7

Number of Pages

1845-1854

Document Type

Article

Personal Identifier

scopus

DOI Link

https://doi.org/10.1016/j.tet.2004.12.015

Socpus ID

19944434175 (Scopus)

Source API URL

https://api.elsevier.com/content/abstract/scopus_id/19944434175

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