Application Of Microphysiological Systems To Enhance Safety Assessment In Drug Discovery
Keywords
drug discovery; microphysiological systems; toxicology
Abstract
Enhancing the early detection of new therapies that are likely to carry a safety liability in the context of the intended patient population would provide a major advance in drug discovery. Microphysiological systems (MPS) technology offers an opportunity to support enhanced preclinical to clinical translation through the generation of higher-quality preclinical physiological data. In this review, we highlight this technological opportunity by focusing on key target organs associated with drug safety and metabolism. By focusing on MPS models that have been developed for these organs, alongside other relevant in vitro models, we review the current state of the art and the challenges that still need to be overcome to ensure application of this technology in enhancing drug discovery.
Publication Date
1-6-2018
Publication Title
Annual Review of Pharmacology and Toxicology
Volume
58
Number of Pages
65-82
Document Type
Article
Personal Identifier
scopus
DOI Link
https://doi.org/10.1146/annurev-pharmtox-010617-052722
Copyright Status
Unknown
Socpus ID
85040620605 (Scopus)
Source API URL
https://api.elsevier.com/content/abstract/scopus_id/85040620605
STARS Citation
Ewart, Lorna; Dehne, Eva Maria; Fabre, Kristin; Gibbs, Susan; and Hickman, James, "Application Of Microphysiological Systems To Enhance Safety Assessment In Drug Discovery" (2018). Scopus Export 2015-2019. 10619.
https://stars.library.ucf.edu/scopus2015/10619